| Synthesis, enzyme kinetics and computational evaluation of N-(β-d-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors M Polyák, G Varga, B Szilágyi, L Juhász, T Docsa, P Gergely, J Begum, ... Bioorganic & medicinal chemistry 21 (18), 5738-5747, 2013 | 32 | 2013 |
| Drug discovery strategies and the preclinical development of D-amino-acid oxidase inhibitors as antipsychotic therapies B Szilágyi, GG Ferenczy, GM Keserű Expert Opinion on Drug Discovery 13 (10), 973-982, 2018 | 12 | 2018 |
| Discovery of isatin and 1H-indazol-3-ol derivatives as d-amino acid oxidase (DAAO) inhibitors B Szilágyi, P Kovács, GG Ferenczy, A Rácz, K Németh, J Visy, P Szabó, ... Bioorganic & Medicinal Chemistry 26 (8), 1579-1587, 2018 | 12 | 2018 |
| Synthesis and characterization of new fluorescent boro-β-carboline dyes DS Kovács, I Hajdu, G Mészáros, L Wittner, D Meszéna, EZ Tóth, ... RSC advances 11 (21), 12802-12807, 2021 | 11 | 2021 |
| Validation of tautomeric and protomeric binding modes by free energy calculations. A case study for the structure based optimization of d-amino acid oxidase … Z Orgován, GG Ferenczy, T Steinbrecher, B Szilágyi, D Bajusz, ... Journal of Computer-Aided Molecular Design 32, 331-345, 2018 | 10 | 2018 |
| Discovery of selective fragment-sized immunoproteasome inhibitors L Kollár, M Gobec, B Szilágyi, M Proj, D Knez, P Ábrányi-Balogh, L Petri, ... European Journal of Medicinal Chemistry 219, 113455, 2021 | 9 | 2021 |
| Discovery of d-amino acid oxidase inhibitors based on virtual screening against the lid-open enzyme conformation B Szilágyi, Ž Skok, A Rácz, GG Ferenczy, J Ilaš, GM Keserű Bioorganic & Medicinal Chemistry Letters 28 (10), 1693-1698, 2018 | 5 | 2018 |
| Synthesis and Biochemical Evaluation of Lid-Open d-Amino Acid Oxidase Inhibitors B Szilágyi, C Hargitai, ÁA Kelemen, A Rácz, GG Ferenczy, B Volk, ... Molecules 24 (2), 290, 2019 | 2 | 2019 |
| Safe and Efficient Continuous-Flow Synthesis and Batchwise Hydrolysis of Ethyl 5-Acetyl-1H-pyrazole-3-carboxylate: A Key Synthon of Darolutamide B Szilágyi, A Egyed, I Mándity, T Nagy, K Kátai-Fadgyas, B Volk, ... Synthesis 55 (06), 959-966, 2023 | 1 | 2023 |
| Design and synthesis of D-amino acid oxidase inhibitors B Szilágyi PQDT-Global, 2019 | | 2019 |
| SAR STUDY OF GLYCOGEN PHOSPHORYLASE INHIBITORS: HETEROCYCLES AS BIOISOSTERIC AMIDE REPLACEMENTS IN N-ACYL-β-D-GLUCOPYRANOSYLAMINES AND N-ACYL-N’-β-DGLUCOPYRANOSYL UREAS B Szilágyi | | |
György M. KeserűHungarian Academy of SciencesVerified email at ttk.mta.hu
