Microwave assisted synthesis: a new technology in drug discovery V Santagada, F Frecentese, E Perissutti, F Fiorino, B Severino, ... Mini reviews in medicinal chemistry 9 (3), 340-358, 2009 | 135 | 2009 |
Anticancer activities of fatty acids and their heterocyclic derivatives M Jóźwiak, A Filipowska, F Fiorino, M Struga European journal of pharmacology 871, 172937, 2020 | 119 | 2020 |
Derivatives as 5HT1A receptor ligands-past and present G Caliendo, V Santagada, E Perissutti, F Fiorino Current medicinal chemistry 12 (15), 1721-1753, 2005 | 115 | 2005 |
5-HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer F Fiorino, B Severino, E Magli, A Ciano, G Caliendo, V Santagada, ... Journal of Medicinal Chemistry 57 (11), 4407-4426, 2014 | 91 | 2014 |
Microwave-enhanced solution coupling of the α, α-dialkyl amino acid, Aib V Santagada, F Fiorino, E Perissutti, B Severino, V De Filippis, B Vivenzio, ... Tetrahedron Letters 42 (31), 5171-5173, 2001 | 65 | 2001 |
Heavy Metals Size Distribution in PM10 and Environmental-Sanitary Risk Analysis in Acerra (Italy) P Di Vaio, E Magli, G Caliendo, A Corvino, F Fiorino, F Frecentese, ... Atmosphere 9 (2), 58, 2018 | 64 | 2018 |
Calpastatin exon 1B-derived peptide, a selective inhibitor of calpain: enhancing cell permeability by conjugation with penetratin S Gil-Parrado, I Assfalg-Machleidt, F Fiorino, D Deluca, D Pfeiler, ... Walter de Gruyter 384 (3), 395-402, 2003 | 62 | 2003 |
Microwave enhanced solution synthesis of 1, 4-benzodiazepin-5-ones V Santagada, E Perissutti, F Fiorino, B Vivenzio, G Caliendo Tetrahedron Letters 42 (12), 2397-2400, 2001 | 59 | 2001 |
Preparation and local anaesthetic activity of benzotriazinone and benzoyltriazole derivatives G Caliendo, F Fiorino, P Grieco, E Perissutti, V Santagada, R Meli, ... European journal of medicinal chemistry 34 (12), 1043-1051, 1999 | 57 | 1999 |
Synthesis and pharmacological evaluations of sildenafil analogues for treatment of erectile dysfunction HA Flores Toque, FBM Priviero, CE Teixeira, E Perissutti, F Fiorino, ... Journal of medicinal chemistry 51 (9), 2807-2815, 2008 | 56 | 2008 |
A convenient synthesis by microwave heating and pharmacological evaluation of novel benzoyltriazole and saccharine derivatives as 5-HT1A receptor ligands G Caliendo, F Fiorino, E Perissutti, B Severino, D Scolaro, S Gessi, ... European journal of pharmaceutical sciences 16 (1-2), 15-28, 2002 | 54 | 2002 |
Trends in H2S-Donors Chemistry and Their Effects in Cardiovascular Diseases A Corvino, F Frecentese, E Magli, E Perissutti, V Santagada, ... Antioxidants 10 (3), 429, 2021 | 53 | 2021 |
Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands G Caliendo, F Fiorino, E Perissutti, B Severino, S Gessi, E Cattabriga, ... European journal of medicinal chemistry 36 (11-12), 873-886, 2001 | 52 | 2001 |
Level, potential sources of polycyclic aromatic hydrocarbons (PAHs) in particulate matter (PM10) in Naples P Di Vaio, B Cocozziello, A Corvino, F Fiorino, F Frecentese, E Magli, ... Atmospheric environment 129, 186-196, 2016 | 51 | 2016 |
Neurounina-1, a novel compound that increases Na+/Ca2+ exchanger activity, effectively protects against stroke damage P Molinaro, M Cantile, O Cuomo, A Secondo, A Pannaccione, ... Molecular Pharmacology 83 (1), 142-156, 2013 | 51 | 2013 |
Synthesis by microwave irradiation of a substituted benzoxazine parallel library with preferential relaxant activity for guinea pig trachealis G Caliendo, E Perissutti, V Santagada, F Fiorino, B Severino, D Cirillo, ... European journal of medicinal chemistry 39 (10), 815-826, 2004 | 50 | 2004 |
1, 2, 4-Thiadiazolidin-3, 5-diones as novel hydrogen sulfide donors B Severino, A Corvino, F Fiorino, P Luciano, F Frecentese, E Magli, ... European Journal of Medicinal Chemistry 143, 1677-1686, 2018 | 45 | 2018 |
New 5-Hydroxytryptamine1A Receptor Ligands Containing a Norbornene Nucleus: Synthesis and in Vitro Pharmacological Evaluation F Fiorino, E Perissutti, B Severino, V Santagada, D Cirillo, S Terracciano, ... Journal of medicinal chemistry 48 (17), 5495-5503, 2005 | 44 | 2005 |
Synthesis and vasorelaxant activity of new 1, 4-benzoxazine derivatives potassium channel openers G Caliendo, E Perissutti, V Santagada, F Fiorino, B Severino, ... Bioorganic & medicinal chemistry 10 (8), 2663-2669, 2002 | 42 | 2002 |
Synthesis of new 1, 2, 3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands G Caliendo, F Fiorino, P Grieco, E Perissutti, V Santagada, B Severino, ... Bioorganic & medicinal chemistry 8 (3), 533-538, 2000 | 42 | 2000 |