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Jorge Esquivias Provencio
Jorge Esquivias Provencio
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Cited by
Year
Structure-Guided Lead Optimization of Triazolopyrimidine-Ring Substituents Identifies Potent Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors …
JM Coteron, M Marco, J Esquivias, X Deng, KL White, J White, M Koltun, ...
Journal of medicinal chemistry 54 (15), 5540-5561, 2011
3202011
A Copper(II)‐Catalyzed Aza‐Friedel–Crafts Reaction of N‐(2‐Pyridyl)sulfonyl Aldimines: Synthesis of Unsymmetrical Diaryl Amines and Triaryl Methanes
J Esquivias, R Gómez Arrayás, JC Carretero
Angewandte Chemie International Edition 45 (4), 629-633, 2006
2572006
Catalytic Asymmetric Inverse-Electron-Demand Diels−Alder Reaction of N-Sulfonyl-1-Aza-1,3-Dienes
J Esquivias, RG Arrayás, JC Carretero
Journal of the American Chemical Society 129 (6), 1480-1481, 2007
2012007
Catalytic asymmetric cross-couplings of racemic α-bromoketones with arylzinc reagents
PM Lundin, J Esquivias, GC Fu
Angewandte Chemie (International ed. in English) 48 (1), 154, 2009
1652009
Tetrahydropyrazolo [1, 5-a] pyrimidine-3-carboxamide and N-benzyl-6′, 7′-dihydrospiro [piperidine-4, 4′-thieno [3, 2-c] pyran] analogues with bactericidal efficacy against …
MJ Remuiñán, E Pérez-Herrán, J Rullás, C Alemparte, M Martínez-Hoyos, ...
PloS one 8 (4), e60933, 2013
1522013
Copper-catalyzed enantioselective conjugate addition of dialkylzinc reagents to (2-pyridyl) sulfonyl imines of chalcones
J Esquivias, RG Arrayás, JC Carretero
The Journal of Organic Chemistry 70 (18), 7451-7454, 2005
992005
Synthesis of nanostructures based on 1, 4-and 1, 3, 5-ethynylphenyl subunits with π-extended conjugation. Carbon dendron units
JG Rodríguez, J Esquivias, A Lafuente, C Díaz
The Journal of Organic Chemistry 68 (21), 8120-8128, 2003
752003
Understanding the Behavior of N-Tosyl and N-2-Pyridylsulfonyl Imines in CuII-Catalyzed Aza-Friedel−Crafts Reactions
I Alonso, J Esquivias, R Gómez-Arrayás, JC Carretero
The Journal of Organic Chemistry 73 (16), 6401-6404, 2008
732008
Inhibiting mycobacterial tryptophan synthase by targeting the inter-subunit interface
KA Abrahams, JAG Cox, K Fütterer, J Rullas, F Ortega-Muro, NJ Loman, ...
Scientific Reports 7 (1), 9430, 2017
572017
Alkylation of Aryl N‐(2‐Pyridylsulfonyl)aldimines with Organozinc Halides: Conciliation of Reactivity and Chemoselectivity
J Esquivias, R Gómez Arrayás, JC Carretero
Angewandte Chemie International Edition 46 (48), 9257-9260, 2007
362007
Novel inhibitors of Mycobacterium tuberculosis GuaB2 identified by a target based high-throughput phenotypic screen
JAG Cox, G Mugumbate, LVG Del Peral, M Jankute, KA Abrahams, ...
Scientific reports 6 (1), 38986, 2016
302016
Easy-To-Synthesize Spirocyclic Compounds Possess Remarkable in Vivo Activity against Mycobacterium tuberculosis
A Guardia, J Baiget, M Cacho, A Pérez, M Ortega-Guerra, W Nxumalo, ...
Journal of Medicinal Chemistry 61 (24), 11327-11340, 2018
252018
Synthesis of conjugated 2 and 2, 5-(ethenyl) and (ethynyl) phenylethynyl thiophenes: fluorescence properties
JG Rodriguez, J Esquivias, A Lafuente, L Rubio
Tetrahedron 62 (13), 3112-3122, 2006
242006
Synthesis of nanostructures based on 1, 4-and 1, 3, 5-phenylethynyl units with π-extended conjugation. Carbon networks dendrimer base units
JG Rodrı́guez, J Esquivias
Tetrahedron letters 44 (26), 4831-4834, 2003
222003
Inverse-Electron-Demand Diels-Alder Reactions of N-(Heteroarylsulfonyl)-1-aza-1, 3-dienes Catalyzed by Chiral Lewis Acids
J Esquivias, I Alonso, RG Arrayas, JC Carretero
Synthesis, 113-126, 2008
202008
Synthesis and optical properties of conjugated N, N-dimethyl and thienyl end-capped 2, 5-(arylethynyl) thiophene oligomer structures
JG Rodrı́guez, A Lafuente, L Rubio, J Esquivias
Tetrahedron letters 45 (38), 7061-7064, 2004
172004
GSK2556286 Is a Novel Antitubercular Drug Candidate Effective In Vivo with the Potential To Shorten Tuberculosis Treatment
EL Nuermberger, MS Martínez-Martínez, O Sanz, B Urones, J Esquivias, ...
Antimicrobial agents and chemotherapy 66 (6), e00132-22, 2022
142022
Exploring the SAR of the β-Ketoacyl-ACP Synthase Inhibitor GSK3011724A and Optimization around a Genotoxic Metabolite
F Cunningham, J Esquivias, R Fernández-Menéndez, A Pérez, A Guardia, ...
ACS Infectious Diseases 6 (5), 1098-1109, 2020
142020
Synthesis of carbon dendron nano-chains with π-extended conjugation based on linear 1, 4-phenylethynyl and 1, 5-naphthylethynyl subunits
JG Rodrı́guez, JL Tejedor, J Esquivias, C Dı́az
Tetrahedron letters 44 (34), 6375-6378, 2003
142003
Tetrahydropyrazolo [1, 5-A] pyrimidine as anti-tuberculosis compounds
E Alvarez-Ruiz, L Ballell-Pages, JC Pichel, L Encinas, J Esquivias, ...
US Patent App. 14/112,564, 2014
82014
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