Structure-Guided Lead Optimization of Triazolopyrimidine-Ring Substituents Identifies Potent Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors … JM Coteron, M Marco, J Esquivias, X Deng, KL White, J White, M Koltun, ... Journal of medicinal chemistry 54 (15), 5540-5561, 2011 | 320 | 2011 |
A Copper(II)‐Catalyzed Aza‐Friedel–Crafts Reaction of N‐(2‐Pyridyl)sulfonyl Aldimines: Synthesis of Unsymmetrical Diaryl Amines and Triaryl Methanes J Esquivias, R Gómez Arrayás, JC Carretero Angewandte Chemie International Edition 45 (4), 629-633, 2006 | 257 | 2006 |
Catalytic Asymmetric Inverse-Electron-Demand Diels−Alder Reaction of N-Sulfonyl-1-Aza-1,3-Dienes J Esquivias, RG Arrayás, JC Carretero Journal of the American Chemical Society 129 (6), 1480-1481, 2007 | 201 | 2007 |
Catalytic asymmetric cross-couplings of racemic α-bromoketones with arylzinc reagents PM Lundin, J Esquivias, GC Fu Angewandte Chemie (International ed. in English) 48 (1), 154, 2009 | 165 | 2009 |
Tetrahydropyrazolo [1, 5-a] pyrimidine-3-carboxamide and N-benzyl-6′, 7′-dihydrospiro [piperidine-4, 4′-thieno [3, 2-c] pyran] analogues with bactericidal efficacy against … MJ Remuiñán, E Pérez-Herrán, J Rullás, C Alemparte, M Martínez-Hoyos, ... PloS one 8 (4), e60933, 2013 | 152 | 2013 |
Copper-catalyzed enantioselective conjugate addition of dialkylzinc reagents to (2-pyridyl) sulfonyl imines of chalcones J Esquivias, RG Arrayás, JC Carretero The Journal of Organic Chemistry 70 (18), 7451-7454, 2005 | 99 | 2005 |
Synthesis of nanostructures based on 1, 4-and 1, 3, 5-ethynylphenyl subunits with π-extended conjugation. Carbon dendron units JG Rodríguez, J Esquivias, A Lafuente, C Díaz The Journal of Organic Chemistry 68 (21), 8120-8128, 2003 | 75 | 2003 |
Understanding the Behavior of N-Tosyl and N-2-Pyridylsulfonyl Imines in CuII-Catalyzed Aza-Friedel−Crafts Reactions I Alonso, J Esquivias, R Gómez-Arrayás, JC Carretero The Journal of Organic Chemistry 73 (16), 6401-6404, 2008 | 73 | 2008 |
Inhibiting mycobacterial tryptophan synthase by targeting the inter-subunit interface KA Abrahams, JAG Cox, K Fütterer, J Rullas, F Ortega-Muro, NJ Loman, ... Scientific Reports 7 (1), 9430, 2017 | 57 | 2017 |
Alkylation of Aryl N‐(2‐Pyridylsulfonyl)aldimines with Organozinc Halides: Conciliation of Reactivity and Chemoselectivity J Esquivias, R Gómez Arrayás, JC Carretero Angewandte Chemie International Edition 46 (48), 9257-9260, 2007 | 36 | 2007 |
Novel inhibitors of Mycobacterium tuberculosis GuaB2 identified by a target based high-throughput phenotypic screen JAG Cox, G Mugumbate, LVG Del Peral, M Jankute, KA Abrahams, ... Scientific reports 6 (1), 38986, 2016 | 30 | 2016 |
Easy-To-Synthesize Spirocyclic Compounds Possess Remarkable in Vivo Activity against Mycobacterium tuberculosis A Guardia, J Baiget, M Cacho, A Pérez, M Ortega-Guerra, W Nxumalo, ... Journal of Medicinal Chemistry 61 (24), 11327-11340, 2018 | 25 | 2018 |
Synthesis of conjugated 2 and 2, 5-(ethenyl) and (ethynyl) phenylethynyl thiophenes: fluorescence properties JG Rodriguez, J Esquivias, A Lafuente, L Rubio Tetrahedron 62 (13), 3112-3122, 2006 | 24 | 2006 |
Synthesis of nanostructures based on 1, 4-and 1, 3, 5-phenylethynyl units with π-extended conjugation. Carbon networks dendrimer base units JG Rodrı́guez, J Esquivias Tetrahedron letters 44 (26), 4831-4834, 2003 | 22 | 2003 |
Inverse-Electron-Demand Diels-Alder Reactions of N-(Heteroarylsulfonyl)-1-aza-1, 3-dienes Catalyzed by Chiral Lewis Acids J Esquivias, I Alonso, RG Arrayas, JC Carretero Synthesis, 113-126, 2008 | 20 | 2008 |
Synthesis and optical properties of conjugated N, N-dimethyl and thienyl end-capped 2, 5-(arylethynyl) thiophene oligomer structures JG Rodrı́guez, A Lafuente, L Rubio, J Esquivias Tetrahedron letters 45 (38), 7061-7064, 2004 | 17 | 2004 |
GSK2556286 Is a Novel Antitubercular Drug Candidate Effective In Vivo with the Potential To Shorten Tuberculosis Treatment EL Nuermberger, MS Martínez-Martínez, O Sanz, B Urones, J Esquivias, ... Antimicrobial agents and chemotherapy 66 (6), e00132-22, 2022 | 14 | 2022 |
Exploring the SAR of the β-Ketoacyl-ACP Synthase Inhibitor GSK3011724A and Optimization around a Genotoxic Metabolite F Cunningham, J Esquivias, R Fernández-Menéndez, A Pérez, A Guardia, ... ACS Infectious Diseases 6 (5), 1098-1109, 2020 | 14 | 2020 |
Synthesis of carbon dendron nano-chains with π-extended conjugation based on linear 1, 4-phenylethynyl and 1, 5-naphthylethynyl subunits JG Rodrı́guez, JL Tejedor, J Esquivias, C Dı́az Tetrahedron letters 44 (34), 6375-6378, 2003 | 14 | 2003 |
Tetrahydropyrazolo [1, 5-A] pyrimidine as anti-tuberculosis compounds E Alvarez-Ruiz, L Ballell-Pages, JC Pichel, L Encinas, J Esquivias, ... US Patent App. 14/112,564, 2014 | 8 | 2014 |