| Computational and biological profile of boronic acids for the detection of bacterial serine-and metallo-β-lactamases M Santucci, F Spyrakis, S Cross, A Quotadamo, D Farina, D Tondi, ... Scientific reports 7 (1), 17716, 2017 | 42 | 2017 |
| Aryl thiosemicarbazones for the treatment of trypanosomatidic infections P Linciano, CB Moraes, LM Alcantara, CH Franco, B Pascoalino, ... European Journal of Medicinal Chemistry 146, 423-434, 2018 | 37 | 2018 |
| X-ray crystallography deciphers the activity of broad-spectrum boronic acid β-lactamase inhibitors L Cendron, A Quotadamo, L Maso, P Bellio, M Montanari, G Celenza, ... ACS Medicinal Chemistry Letters 10 (4), 650-655, 2019 | 28 | 2019 |
| Enhancement of benzothiazoles as pteridine reductase-1 inhibitors for the treatment of trypanosomatidic infections P Linciano, C Pozzi, LD Iacono, F di Pisa, G Landi, A Bonucci, S Gul, ... Journal of Medicinal Chemistry 62 (8), 3989-4012, 2019 | 27 | 2019 |
| Comparative mapping of on-targets and off-targets for the discovery of anti-trypanosomatid folate pathway inhibitors J Panecka-Hofman, I Pöhner, F Spyrakis, T Zeppelin, F Di Pisa, LD Iacono, ... Biochimica et Biophysica Acta (BBA)-General Subjects 1861 (12), 3215-3230, 2017 | 25 | 2017 |
| Accelerating drug discovery efforts for trypanosomatidic infections using an integrated transnational academic drug discovery platform CB Moraes, G Witt, M Kuzikov, B Ellinger, T Calogeropoulou, KC Prousis, ... SLAS DISCOVERY: Advancing Life Sciences R&D 24 (3), 346-361, 2019 | 22 | 2019 |
| Human thymidylate synthase inhibitors halting ovarian cancer growth S Ferrari, L Severi, C Pozzi, A Quotadamo, G Ponterini, L Losi, G Marverti, ... Vitamins and Hormones 107, 473-513, 2018 | 18 | 2018 |
| An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases A Quotadamo, P Linciano, P Davoli, D Tondi, MP Costi, A Venturelli Synlett 27 (17), 2447-2450, 2016 | 15 | 2016 |
| Multitarget, selective compound design yields potent inhibitors of a kinetoplastid pteridine reductase 1 I Pöhner, A Quotadamo, J Panecka-Hofman, R Luciani, M Santucci, ... Journal of Medicinal Chemistry 65 (13), 9011-9033, 2022 | 11 | 2022 |
| First virtual screening and experimental validation of inhibitors targeting GES-5 carbapenemase F Spyrakis, P Bellio, A Quotadamo, P Linciano, P Benedetti, G D’Arrigo, ... Journal of computer-aided molecular design 33, 295-305, 2019 | 9 | 2019 |
| Scaffolds and biological targets avenue to fight against drug resistance in leishmaniasis C Borsari, A Quotadamo, S Ferrari, A Venturelli, A Cordeiro-da-Silva, ... Annual Reports in Medicinal Chemistry 51, 39-95, 2018 | 8 | 2018 |
| New Insights into Bioactive Compounds from the Medicinal Plant Spathodea campanulata P. Beauv. and Their Activity against Helicobacter pylori CR Ngnameko, L Marchetti, B Zambelli, A Quotadamo, D Roncarati, ... Antibiotics 9 (5), 258, 2020 | 6 | 2020 |
| Diastereoselective Synthesis of (1, 3‐Dioxan‐4‐yl) pyrimidine and Purin Nucleoside Analogues UM Battisti, C Sorbi, A Quotadamo, S Franchini, A Tait, D Schols, ... European Journal of Organic Chemistry 2015 (6), 1235-1245, 2015 | 5 | 2015 |
| Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth L Costantino, S Ferrari, M Santucci, OMH Salo-Ahen, E Carosati, ... Elife 11, e73862, 2022 | 4 | 2022 |
| Structure–Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis M Dichiara, QJ Simpson, A Quotadamo, HB Jalani, AX Huang, CC Millard, ... ACS Infectious Diseases 9 (8), 1470-1487, 2023 | 3 | 2023 |
| Optimization of N‐alkylation in the Synthesis of Methotrexate and Pteridine‐based Derivatives Under Microwave‐Irradiation A Quotadamo, P Linciano, MP Costi, A Venturelli ChemistrySelect 4 (15), 4429-4433, 2019 | 3 | 2019 |
| Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes L Ferrins, MJ Buskes, MM Kapteyn, HN Engels, SE Enos, C Lu, DM Klug, ... Frontiers in Microbiology 14, 1149145, 2023 | 2 | 2023 |
| Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus DM Klug, EG Tse, DG Silva, Y Cao, SA Charman, J Chauhan, E Crighton, ... ACS Infectious Diseases 9 (12), 2423-2435, 2023 | 1 | 2023 |
| High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic Agents P Linciano, A Quotadamo, R Luciani, M Santucci, KM Zorn, DH Foil, ... Journal of Medicinal Chemistry 66 (22), 15230-15255, 2023 | 1 | 2023 |
| Disrupters of the Thymidylate Synthase Homodimer Accelerate Its Proteasomal Degradation and Inhibit Cancer Growth. C Luca, S Ferrari, M Santucci, OM Salo-Ahen, C Emanuele, S Franchini, ... | 1 | 2021 |
