| Linker-modified quinoline derivatives targeting HIV-1 integrase: synthesis and biological activity C Bénard, F Zouhiri, M Normand-Bayle, M Danet, D Desmaële, H Leh, ... Bioorganic & medicinal chemistry letters 14 (10), 2473-2476, 2004 | 143 | 2004 |
| HIV-1 replication inhibitors of the styrylquinoline class: Introduction of an additional carboxyl group at the C-5 position of the quinoline F Zouhiri, M Danet, C Bénard, M Normand-Bayle, JF Mouscadet, H Leh, ... Tetrahedron Letters 46 (13), 2201-2205, 2005 | 124 | 2005 |
| Reaction of rosmarinic acid with nitrite ions in acidic conditions: discovery of nitro-and dinitrorosmarinic acids as new anti-HIV-1 agents M Dubois, F Bailly, G Mbemba, JF Mouscadet, Z Debyser, M Witvrouw, ... Journal of medicinal chemistry 51 (8), 2575-2579, 2008 | 96 | 2008 |
| New HIV-1 replication inhibitors of the styryquinoline class bearing aroyl/acyl groups at the C-7 position: synthesis and biological activity M Normand-Bayle, C Bénard, F Zouhiri, JF Mouscadet, H Leh, ... Bioorganic & medicinal chemistry letters 15 (18), 4019-4022, 2005 | 80 | 2005 |
| Inhibition of early steps of HIV-1 replication by SNF5/Ini1 M Maroun, O Delelis, G Coadou, T Bader, E Ségéral, G Mbemba, C Petit, ... Journal of biological chemistry 281 (32), 22736-22743, 2006 | 74 | 2006 |
| Spectroscopic studies of diketoacids− metal interactions. A probing tool for the pharmacophoric intermetallic distance in the HIV-1 integrase active site C Maurin, F Bailly, E Buisine, H Vezin, G Mbemba, JF Mouscadet, ... Journal of medicinal chemistry 47 (22), 5583-5586, 2004 | 61 | 2004 |
| Synthesis and HIV-1 integrase inhibitory activities of caffeic acid dimers derived from Salvia officinalis F Bailly, C Queffelec, G Mbemba, JF Mouscadet, P Cotelle Bioorganic & Medicinal Chemistry Letters 15 (22), 5053-5056, 2005 | 54 | 2005 |
| Efficient and specific internal cleavage of a retroviral palindromic DNA sequence by tetrameric HIV-1 integrase O Delelis, V Parissi, H Leh, G Mbemba, C Petit, P Sonigo, E Deprez, ... PloS one 2 (7), e608, 2007 | 51 | 2007 |
| Synthesis and biological activities of a series of 4, 5-diaryl-3-hydroxy-2 (5H)-furanones F Bailly, C Queffélec, G Mbemba, JF Mouscadet, N Pommery, J Pommery, ... European journal of medicinal chemistry 43 (6), 1222-1229, 2008 | 39 | 2008 |
| Synthesis and antiviral properties of some polyphenols related to Salvia genus C Queffélec, F Bailly, G Mbemba, JF Mouscadet, S Hayes, Z Debyser, ... Bioorganic & medicinal chemistry letters 18 (16), 4736-4740, 2008 | 38 | 2008 |
| A novel function for spumaretrovirus integrase: an early requirement for integrase-mediated cleavage of 2 LTR circles O Delelis, C Petit, H Leh, G Mbemba, JF Mouscadet, P Sonigo Retrovirology 2, 1-18, 2005 | 36 | 2005 |
| Design, synthesis, and anti-integrase activity of catechol–DKA hybrids C Maurin, F Bailly, G Mbemba, JF Mouscadet, P Cotelle Bioorganic & medicinal chemistry 14 (9), 2978-2984, 2006 | 33 | 2006 |
| Synthesis, biological evaluation and molecular modeling studies of quinolonyl diketo acid derivatives: new structural insight into the HIV-1 integrase inhibition P Vandurm, A Guiguen, C Cauvin, B Georges, K Le Van, C Michaux, ... European journal of medicinal chemistry 46 (5), 1749-1756, 2011 | 32 | 2011 |
| New 2-arylnaphthalenediols and triol inhibitors of HIV-1 integrase—Discovery of a new polyhydroxylated antiviral agent C Maurin, C Lion, F Bailly, N Touati, H Vezin, G Mbemba, JF Mouscadet, ... Bioorganic & medicinal chemistry 18 (14), 5194-5201, 2010 | 16 | 2010 |
| Structural and theoretical studies of [6-bromo-1-(4-fluorophenylmethyl)-4(1H)-quinolinon-3-yl)]-4-hydroxy-2-oxo-3-butenoïc acid as HIV-1 integrase inhibitor P Vandurm, C Cauvin, A Guiguen, B Georges, K Le Van, V Martinelli, ... Bioorganic & medicinal chemistry letters 19 (16), 4806-4809, 2009 | 14 | 2009 |
| The total synthesis of fukiic acid, an HIV-1 integrase inhibitor C Queffélec, F Bailly, G Mbemba, JF Mouscadet, Z Debyser, M Witvrouw, ... European journal of medicinal chemistry 43 (10), 2268-2271, 2008 | 10 | 2008 |
| Synthesis and anti-HIV-1 integrase activity of modified dinucleotides Y Aubert, M Chassignol, V Roig, G Mbemba, J Weiss, H Meudal, ... European journal of medicinal chemistry 44 (12), 5029-5044, 2009 | 9 | 2009 |
| Biochemical properties of the xenotropic murine leukemia virus-related virus integrase G Mbemba, E Henry, O Delelis, MC Bouger, M Buckle, JF Mouscadet, ... Biochimie 107, 300-309, 2014 | | 2014 |
| HIV-1 integrase inhibition by quinolone compounds: contribution to the rational design of new inhibitors A Guiguen, P Vandurm, C Cauvin, B George, K Le Van, V Martinelli, ... Abstract of Forum de recherches fondamentales et cliniques sur le VIH, 2010 | | 2010 |
| Une nouvelle famille d’inhibiteurs mixtes chélatants de l’intégrase et de la Ribonucléase H du VIH-1: les dérivés de la N-hydroxyisoquinoléine-1, 3-dione. M Billamboz, F Bailly, G Mbemba, JF Mouscadet, A Faure, ML Andréola, ... Semaine d’Etudes de Chimie Organique (SECO45), 2008 | | 2008 |
